Drug Standards
![Medchemexpress LLC Hexanoic acid, 6-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1-oxo-1H-isoindol-4-yl]amino]- | 2338824-30-7 | 96.4% | 373.40 | 25 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/default.jpg-250.jpg)
Medchemexpress LLC Hexanoic acid, 6-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1-oxo-1H-isoindol-4-yl]amino]- | 2338824-30-7 | 96.4% | 373.40 | 25 MG
Lenalidomide-C5-acid is a Lenalidomide-based E3 ligase ligand-linker conjugate utilized in the recruitment of CRBN protein, and it can be used to synthesize PROTACs. The product is for research use only and not sold to patients.
- Lenalidomide-based E3 ligase ligand-linker conjugate
- Used in the recruitment of CRBN protein
- Can be used to synthesize PROTACs
- Appearance: Solid
- Color: Off-white to light yellow
Medchemexpress LLC Lenalidomide 4'-PEG1-amine dihydrochloride | 2624336-86-1 | 98.37% | 419.30 | 5 MG
Lenalidomide 4'-PEG1-amine dihydrochloride is a Lenalidomide-based Cereblon ligand used in the recruitment of CRBN protein. It can be connected to the ligand for protein by a linker to form PROTAC.
- Lenalidomide-based Cereblon ligand
- Used in the recruitment of CRBN protein
- Can be connected to the ligand for protein by a linker to form PROTAC
- For research use only
Medchemexpress LLC Lenalidomide 4'-PEG2-amine dihydrochloride | 2624336-88-3 | 99.0% | 463.36 | 1 ML
Lenalidomide 4'-PEG2-amine dihydrochloride is a Lenalidomide-based Cereblon ligand that plays a role in the recruitment of CRBN protein. It can be connected to a ligand for protein by a linker to form PROTAC.
- Functions as a Lenalidomide-based Cereblon ligand.
- Recruits CRBN protein.
- Connects to ligands for protein via a linker to form PROTACs.
Medchemexpress LLC ARQ 621 | 1095253-39-6 | ≥99.0% | 552.43 | 25 MG
ARQ 621 is an allosteric, potent, and selective inhibitor of Eg5, a microtubule-based ATPase motor protein involved in cell division. It exhibits anti-tumor activity and is a kinesin inhibitor. Additionally, ARQ 621 is a click chemistry reagent containing an Alkyne group, capable of undergoing copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
- Allosteric, potent, and selective inhibitor of Eg5
- Microtubule-based ATPase motor protein inhibitor
- Involved in cell division
- Anti-tumor activity
- Kinesin inhibitor
- Click chemistry reagent with an alkyne group
- Undergoes copper-catalyzed azide-alkyne cycloaddition (CuAAc) with azide groups
Medchemexpress LLC Fenoldopam mesylate | 67227-57-0 | 99.9% | 100 MG
Fenoldopam mesylate functions as a D1 receptor agonist and a novel lysine-specific demethylase 1 (LSD1) inhibitor with an IC50 of 0.8974 μM. This compound demonstrates anti-hypertensive effects, exhibits anti-cancer cell proliferation activity, and can induce cell apoptosis, making it a subject of research in various biological contexts.
- Functions as a D1 receptor agonist
- Acts as a novel LSD1 inhibitor
- Exhibits anti-hypertensive properties
- Shows anti-cancer cell proliferation activity
- Capable of inducing cell apoptosis
- Active against RCC cell lines (786-O, ACHN) in vitro
Medchemexpress LLC Fenticonazole Nitrate | 73151-29-8 | 98.9% | 1 ML
Fenticonazole Nitrate is an antifungal imidazole ring derivative. It functions by hindering ergosterol integration, which in turn destructs the cytoplasmatic outer membrane. Fenticonazole Nitrate is effective against Gram-positive bacteria, mycoses, and vaginal candidiasis.
- Antifungal imidazole ring derivative
- Hinders ergosterol integration
- Destroys the cytoplasmatic outer membrane
- Effective against Gram-positive bacteria
- Effective against mycoses
- Effective against vaginal candidiasis
Medchemexpress LLC Diclazuril | 101831-37-2 | 99.7% | 500 MG
Diclazuril is a benzeneacetonitrile derivative and a potent, orally active anticoccidial agent. It is used for research into infectious and parasitic diseases such as coccidiosis, acute toxoplasmosis, and equine protozoal pyoencephalitis (EPM).
- Potent and orally active anticoccidial agent
- Used for research into infectious and parasitic diseases, including coccidiosis, acute toxoplasmosis, and equine protozoal pyoencephalitis (EPM)
- Effective against *E. maxima* later in its life cycle
- Reduces lesion scores and improves performance and health in challenged birds
- Soluble in DMSO at 25 mg/mL (61.33 mM)
Medchemexpress LLC Benzamide, 3-(aminosulfonyl)-4-chloro-N-(2,3-dihydro-2-methyl-1H-indol-1-yl)- | 26807-65-8 | 99.6% | 1 G
Indapamide is an orally active sulphonamide diuretic agent that reduces blood pressure by decreasing vascular reactivity and peripheral vascular resistance. It can also reduce left ventricular hypertrophy.
- Orally active sulphonamide diuretic agent
- Reduces blood pressure by decreasing vascular reactivity and peripheral vascular resistance
- Can reduce left ventricular hypertrophy
- High purity of 99.6%
- Appears as a white to off-white solid
- Soluble in DMSO (≥ 100 mg/mL)
- Demonstrates biological activity in vitro, including reducing insulin secretory response and increasing osteoblast proliferation
- Shown to lower blood pressure in spontaneously hypertensive rats in vivo
Medchemexpress LLC Meloxicam (Standard) | 71125-38-7 | 99.89% | 100 MG
Meloxicam (Standard) is the analytical standard of Meloxicam, intended for research and analytical applications. Meloxicam is a non-steroidal anti-inflammatory agent that inhibits COX activity, with IC50s of 0.49 μM for COX-2 and 36.6 μM for COX-1.
- Intended for research and analytical applications
- Non-steroidal anti-inflammatory agent
- Inhibits COX activity
- Used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS
Medchemexpress LLC Ritodrine hydrochloride | 23239-51-2 | 98.5% | 1 ML
Ritodrine hydrochloride is a potent and orally active β-adrenergic agonist. It is known to decrease preterm delivery and uterine contraction, making it a valuable compound for research into preterm labor.
- Potent and orally active beta-adrenergic agonist
- Decreases preterm delivery
- Decreases uterine contraction
- Potential for research of preterm labor
- Targets beta adrenergic receptor
Medchemexpress LLC Venlafaxine-d6 hydrochloride | 1062606-12-5 | 98.2% | 5 MG
Venlafaxine-d6 hydrochloride is the deuterium labeled Venlafaxine hydrochloride. It is an orally active, potent serotonin (5-HT)/norepinephrine (NE) reuptake dual inhibitor and an antidepressant. It is intended for research purposes only.
- Deuterium labeled compound
- Orally active, potent serotonin (5-HT)/norepinephrine (NE) reuptake dual inhibitor
- Antidepressant
- Used for research purposes only
- Suitable as a tracer for quantitative analysis
- Can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS
Medchemexpress LLC Oxfendazole | 53716-50-0 | MFCD00801063 | 98.8% | 1 G
Oxfendazole is a sulfoxide form of fenbendazole that is effective when taken orally. It fights parasites and has tumor-promoting activity.
- Appearance: White to off-white solid
- Purity: 98.8% (LCMS)
- Molecular Weight: 315.35
- Molecular Formula: C15H13N3O3S
- Consistent with structure by 1H NMR and LCMS
- Intended for laboratory chemicals and substance manufacturing
- For research use only
Medchemexpress LLC Diphenhydramine hydrochloride | 147-24-0 | 99.9% | 1 ML
Diphenhydramine hydrochloride is a first-generation histamine H1-receptor antagonist with anti-cholinergic effects, capable of crossing the ovine blood-brain barrier.
- Acts as a first-generation histamine H1-receptor antagonist
- Exhibits anti-cholinergic effects
- Can cross the ovine blood-brain barrier
- Inhibits cisplatin-induced cell death in kidney cells
- Induces apoptosis in certain cell lines
- Reduces mortality in rats exposed to dichlorvos
Medchemexpress LLC Meloxicam | 71125-38-7 | 99.9% | 50 MG
Meloxicam (Standard) is the analytical standard of Meloxicam. This product is intended for research and analytical applications. Meloxicam is a non-steroidal antiinflammatory agent that inhibits COX activity, with IC50s of 0.49 μM and 36.6 μM for COX-2 and COX-1, respectively. It is commonly used in qualitative, quantitative, and methodological research experiments in HPLC, GC, and MS.
- Analytical standard for Meloxicam
- Intended for research and analytical applications
- Inhibits COX activity
- Used in qualitative, quantitative, and methodological research experiments in HPLC, GC, and MS
Medchemexpress LLC Sarafloxacin hydrochloride | 91296-87-6 | 98.1% | 1 G
Sarafloxacin hydrochloride is a quinolone antibiotic agent, specifically a fluoroquinolone, registered for use in treating poultry diseases. It has demonstrated efficacy in field trials for treating channel catfish infected with E. ictaluri.
- Quinolone antibiotic agent.
- Fluoroquinolone antibiotic.
- Efficacious in treating channel catfish infected with E. ictaluri.